Sfoglia per Autore
The aldol addition of readily enolizable 1,3-dicarbonyl compounds to 2-cyanobenzaldehyde in the synthesis of novel 3-substituted isoindolinones
2011-01-01 More, V.; Dimola, A.; Perillo, M.; Decaprariis, P.; Filosa, R.; Peduto, A.; Massa, A.
Synthesis and reactivity of the 3-substituted isoindolinone framework to assemble highly functionalized related structures
2012-01-01 Petronzi, C.; Collarile, S.; Croce, G.; Filosa, R.; De Caprariis, P.; Peduto, A.; Palombi, L.; Intintoli, V.; Di Mola, A.; Massa, A.
Active methylene compounds in a very effective approach to 3-substituted isobenzofuranones through tandem aldol/lactonization reactions
2012-01-01 Di Mola, A.; Croce, G.; More, V.; De Caprariis, P.; Filosa, R.; Massa, A.
1-methoxy-canthin-6-one and related β-carbolines: From natural compound to synthesis and biological activities
2012-01-01 Peduto, A.; Filosa, R.; De Caprariis, P.; De Feo, V.; Li, S.; Wang, P.; De Martino, L.
Potent inhibition of human 5-lipoxygenase and microsomal prostaglandin E2 synthase-1 by the anti-carcinogenic and anti-inflammatory agent embelin
2013-01-01 Schaible, A. M.; Traber, H.; Temml, V.; Noha, S. M.; Filosa, R.; Peduto, A.; Weinigel, C.; Barz, D.; Schuster, D.; Werz, O.
Cyclohexa-2,5-diene-1,4-dione-based antiproliferative agents: Design, synthesis, and cytotoxic evaluation
2013-01-01 Petronzi, C.; Festa, M.; Peduto, A.; Castellano, M.; Marinello, J.; Massa, A.; Capasso, A.; Capranico, G.; La Gatta, A.; De Rosa, M.; Caraglia, M.; Filosa, R.
Discovery and biological evaluation of novel 1,4-benzoquinone and related resorcinol derivatives that inhibit 5-lipoxygenase
2013-01-01 Filosa, R.; Peduto, A.; Aparoy, P.; Schaible, A. M.; Luderer, S.; Krauth, V.; Petronzi, C.; Massa, A.; De Rosa, M.; Reddanna, P.; Werz, O.
Design of inhibitors of influenza virus membrane fusion: Synthesis, structure-activity relationship and in vitro antiviral activity of a novel indole series
2013-01-01 Brancato, V.; Peduto, A.; Wharton, S.; Martin, S.; More, V.; Di Mola, A.; Massa, A.; Perfetto, B.; Donnarumma, G.; Schiraldi, C.; Tufano, M. A.; de Rosa, M.; Filosa, R.; Hay, A.
Further studies on ethyl 5-hydroxy-indole-3-carboxylate scaffold: Design, synthesis and evaluation of 2-phenylthiomethyl-indole derivatives as efficient inhibitors of human 5-lipoxygenase
2014-01-01 Peduto, A.; Bruno, F.; Dehm, F.; Krauth, V.; De Caprariis, P.; Weinigel, C.; Barz, D.; Massa, A.; De Rosa, M.; Werz, O.; Filosa, R.
Elucidation of the molecular mechanism and the efficacy in vivo of a novel 1,4-benzoquinone that inhibits 5-lipoxygenase
2014-01-01 Schaible, A. M.; Filosa, R.; Temml, V.; Krauth, V.; Matteis, M.; Peduto, A.; Bruno, F.; Luderer, S.; Roviezzo, F.; Di Mola, A.; De Rosa, M.; D'Agostino, B.; Weinigel, C.; Barz, D.; Koeberle, A.; Pergola, C.; Schuster, D.; Werz, O.
Cascade reactions of glycine Schiff bases and chiral phase transfer catalysts in the synthesis of α-amino acids 3-substituted phthalides or isoindolinones
2014-01-01 Perillo, M.; Di Mola, A.; Filosa, R.; Palombi, L.; Massa, A.
In vitro antiviral and immunomodulatory activity of arbidol and structurally related derivatives in herpes simplex virus type 1-infected human keratinocytes (HaCat)
2014-01-01 Perfetto, B.; Filosa, R.; Gregorio, V. D.; Peduto, A.; Gatta, A. L.; Caprariis, P. D.; Tufano, M. A.; Donnarumma, G.
New chelating agents for Cu(II), Fe(III), Al(III), and Zn(II) based on β-diketonate-3-substituted phthalide (isobenzofuranone) and isoindolinone
2014-01-01 Di Matteo, L.; Christodoulakis, O.; Filosa, R.; De Caprariis, P.; Di Mola, A.; Vasca, E.; Massa, A.
Structure-activity relationship study of arbidol derivatives as inhibitors of chikungunya virus replication
2014-01-01 Di Mola, A.; Peduto, A.; La Gatta, A.; Delang, L.; Pastorino, B.; Neyts, J.; Leyssen, P.; De Rosa, M.; Filosa, R.
3-Carboxylate-Substituted Isoindolinones in K2CO3-Catalyzed Michael Reactions
2015-01-01 Scorzelli, F.; Di Mola, A.; Palombi, L.; Filosa, R.; Massa, A.
Novel series of benzoquinones with high potency against 5-lipoxygenase in human polymorphonuclear leukocytes
2015-01-01 Filosa, R.; Peduto, A.; Schaible, A. M.; Krauth, V.; Weinigel, C.; Barz, D.; Petronzi, C.; Bruno, F.; Roviezzo, F.; Spaziano, G.; D'Agostino, B.; De Rosa, M.; Werz, O.
Bifunctional phase-transfer catalysis in the asymmetric synthesis of biologically active isoindolinones
2015-01-01 Di Mola, A.; Tiffner, M.; Scorzelli, F.; Palombi, L.; Filosa, R.; De Caprariis, P.; Waser, M.; Massa, A.
The introduction of inversion of polarity sites in DNA G-quadruplex structures: Effects and perspectives
2016-01-01 Virgilio, A.; Esposito, V.; Filosa, R.; Mayol, L.; Galeone, A.
Role of adiponectin in sphingosine-1-phosphate induced airway hyperresponsiveness and inflammation
2016-01-01 Nigro, E.; Matteis, M.; Roviezzo, F.; Mattera Iacono, V.; Scudiero, O.; Spaziano, G.; Tartaglione, G.; Urbanek, K.; Filosa, R.; Daniele, A.; D'Agostino, B.
Synthesis and pharmacological evaluation of functionalized isoindolinones on GABA-activated chloride currents in rat cerebellum granule cells in culture
2016-01-01 Di Mola, A.; Gatta, E.; Petronzi, C.; Cupello, A.; De Caprariis, P.; Robello, M.; Massa, A.; Filosa, R.
Titolo | Data di pubblicazione | Autore(i) | File |
---|---|---|---|
The aldol addition of readily enolizable 1,3-dicarbonyl compounds to 2-cyanobenzaldehyde in the synthesis of novel 3-substituted isoindolinones | 1-gen-2011 | More, V.; Dimola, A.; Perillo, M.; Decaprariis, P.; Filosa, R.; Peduto, A.; Massa, A. | |
Synthesis and reactivity of the 3-substituted isoindolinone framework to assemble highly functionalized related structures | 1-gen-2012 | Petronzi, C.; Collarile, S.; Croce, G.; Filosa, R.; De Caprariis, P.; Peduto, A.; Palombi, L.; Intintoli, V.; Di Mola, A.; Massa, A. | |
Active methylene compounds in a very effective approach to 3-substituted isobenzofuranones through tandem aldol/lactonization reactions | 1-gen-2012 | Di Mola, A.; Croce, G.; More, V.; De Caprariis, P.; Filosa, R.; Massa, A. | |
1-methoxy-canthin-6-one and related β-carbolines: From natural compound to synthesis and biological activities | 1-gen-2012 | Peduto, A.; Filosa, R.; De Caprariis, P.; De Feo, V.; Li, S.; Wang, P.; De Martino, L. | |
Potent inhibition of human 5-lipoxygenase and microsomal prostaglandin E2 synthase-1 by the anti-carcinogenic and anti-inflammatory agent embelin | 1-gen-2013 | Schaible, A. M.; Traber, H.; Temml, V.; Noha, S. M.; Filosa, R.; Peduto, A.; Weinigel, C.; Barz, D.; Schuster, D.; Werz, O. | |
Cyclohexa-2,5-diene-1,4-dione-based antiproliferative agents: Design, synthesis, and cytotoxic evaluation | 1-gen-2013 | Petronzi, C.; Festa, M.; Peduto, A.; Castellano, M.; Marinello, J.; Massa, A.; Capasso, A.; Capranico, G.; La Gatta, A.; De Rosa, M.; Caraglia, M.; Filosa, R. | |
Discovery and biological evaluation of novel 1,4-benzoquinone and related resorcinol derivatives that inhibit 5-lipoxygenase | 1-gen-2013 | Filosa, R.; Peduto, A.; Aparoy, P.; Schaible, A. M.; Luderer, S.; Krauth, V.; Petronzi, C.; Massa, A.; De Rosa, M.; Reddanna, P.; Werz, O. | |
Design of inhibitors of influenza virus membrane fusion: Synthesis, structure-activity relationship and in vitro antiviral activity of a novel indole series | 1-gen-2013 | Brancato, V.; Peduto, A.; Wharton, S.; Martin, S.; More, V.; Di Mola, A.; Massa, A.; Perfetto, B.; Donnarumma, G.; Schiraldi, C.; Tufano, M. A.; de Rosa, M.; Filosa, R.; Hay, A. | |
Further studies on ethyl 5-hydroxy-indole-3-carboxylate scaffold: Design, synthesis and evaluation of 2-phenylthiomethyl-indole derivatives as efficient inhibitors of human 5-lipoxygenase | 1-gen-2014 | Peduto, A.; Bruno, F.; Dehm, F.; Krauth, V.; De Caprariis, P.; Weinigel, C.; Barz, D.; Massa, A.; De Rosa, M.; Werz, O.; Filosa, R. | |
Elucidation of the molecular mechanism and the efficacy in vivo of a novel 1,4-benzoquinone that inhibits 5-lipoxygenase | 1-gen-2014 | Schaible, A. M.; Filosa, R.; Temml, V.; Krauth, V.; Matteis, M.; Peduto, A.; Bruno, F.; Luderer, S.; Roviezzo, F.; Di Mola, A.; De Rosa, M.; D'Agostino, B.; Weinigel, C.; Barz, D.; Koeberle, A.; Pergola, C.; Schuster, D.; Werz, O. | |
Cascade reactions of glycine Schiff bases and chiral phase transfer catalysts in the synthesis of α-amino acids 3-substituted phthalides or isoindolinones | 1-gen-2014 | Perillo, M.; Di Mola, A.; Filosa, R.; Palombi, L.; Massa, A. | |
In vitro antiviral and immunomodulatory activity of arbidol and structurally related derivatives in herpes simplex virus type 1-infected human keratinocytes (HaCat) | 1-gen-2014 | Perfetto, B.; Filosa, R.; Gregorio, V. D.; Peduto, A.; Gatta, A. L.; Caprariis, P. D.; Tufano, M. A.; Donnarumma, G. | |
New chelating agents for Cu(II), Fe(III), Al(III), and Zn(II) based on β-diketonate-3-substituted phthalide (isobenzofuranone) and isoindolinone | 1-gen-2014 | Di Matteo, L.; Christodoulakis, O.; Filosa, R.; De Caprariis, P.; Di Mola, A.; Vasca, E.; Massa, A. | |
Structure-activity relationship study of arbidol derivatives as inhibitors of chikungunya virus replication | 1-gen-2014 | Di Mola, A.; Peduto, A.; La Gatta, A.; Delang, L.; Pastorino, B.; Neyts, J.; Leyssen, P.; De Rosa, M.; Filosa, R. | |
3-Carboxylate-Substituted Isoindolinones in K2CO3-Catalyzed Michael Reactions | 1-gen-2015 | Scorzelli, F.; Di Mola, A.; Palombi, L.; Filosa, R.; Massa, A. | |
Novel series of benzoquinones with high potency against 5-lipoxygenase in human polymorphonuclear leukocytes | 1-gen-2015 | Filosa, R.; Peduto, A.; Schaible, A. M.; Krauth, V.; Weinigel, C.; Barz, D.; Petronzi, C.; Bruno, F.; Roviezzo, F.; Spaziano, G.; D'Agostino, B.; De Rosa, M.; Werz, O. | |
Bifunctional phase-transfer catalysis in the asymmetric synthesis of biologically active isoindolinones | 1-gen-2015 | Di Mola, A.; Tiffner, M.; Scorzelli, F.; Palombi, L.; Filosa, R.; De Caprariis, P.; Waser, M.; Massa, A. | |
The introduction of inversion of polarity sites in DNA G-quadruplex structures: Effects and perspectives | 1-gen-2016 | Virgilio, A.; Esposito, V.; Filosa, R.; Mayol, L.; Galeone, A. | |
Role of adiponectin in sphingosine-1-phosphate induced airway hyperresponsiveness and inflammation | 1-gen-2016 | Nigro, E.; Matteis, M.; Roviezzo, F.; Mattera Iacono, V.; Scudiero, O.; Spaziano, G.; Tartaglione, G.; Urbanek, K.; Filosa, R.; Daniele, A.; D'Agostino, B. | |
Synthesis and pharmacological evaluation of functionalized isoindolinones on GABA-activated chloride currents in rat cerebellum granule cells in culture | 1-gen-2016 | Di Mola, A.; Gatta, E.; Petronzi, C.; Cupello, A.; De Caprariis, P.; Robello, M.; Massa, A.; Filosa, R. |
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