Sfoglia per Autore  FILOSA, Rosanna

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Mostrati risultati da 1 a 20 di 91
Titolo Data di pubblicazione Autore(i) File
N, N′ (4,5-dihydro-1H-imidazol-2-yl)3-aza-1,10-decane-diamine and N, N′(4,5-dihydro-1H-imidazol-2-yl)3-aza-1, 10-dodecane-diamine antagonize cell proliferation as selective ligands towards topoisomerase II 1-gen-2006 Filosa, R.; Buonerba, M.; Loddo, R.; Busonera, B.; La Colla, P.; Saturnino, C.
Synthesis and biological evaluation of (2S)- and (2R)-2-(3′-phosphonobicyclo[1.1.1]pentyl)glycines as novel group III selective metabotropic glutamate receptor ligands 1-gen-2006 Filosa, R.; Marinozzi, M.; Costantino, G.; Hermit, M. B.; Thomsen, C.; Pellicciari, R.
Synthesis and preliminary biological evaluation of 2′-substituted 2-(3′-carboxybicyclo[1.1.1]-pentyl)glycine derivatives as group I selective metabotropic glutamate receptor ligands 1-gen-2006 Pellicciari, R.; Filosa, R.; Fulco, M. C.; Marinozzi, M.; Macchiarulo, A.; Novak, C.; Natalini, B.; Hermit, M. B.; Nielsen, S.; Sager, T. N.; Stensbol, T. B.; Thomsen, C.
Evaluation of alternative strategies to optimize ketorolac transdermal delivery 1-gen-2006 Puglia, C; Filosa, R; Peduto, A; de Caprariis, P; Rizza, L; Bonina, F; Blasi, P
Diastereoselectivity in the alkylation of 4-fluoroproline methyl esters 1-gen-2006 Filosa, R.; Holder, C.; Auberson, Y. P.
Synthesis and antiproliferative properties of N3/8-disubstituted 3,8-diazabicyclo[3.2.1]octane analogues of 3,8-bis[2-(3,4,5-trimethoxyphenyl)pyridin-4-yl]methyl-piperazine 1-gen-2007 Filosa, R.; Peduto, A.; de Caprariis, P.; Saturnino, C.; Festa, M.; Petrella, A.; Pau, A.; Pinna, G. A.; La Colla, P.; Busonera, B.; Loddo, R.
Synthesis, physicochemical properties and in vitro permeation studies of new ketorolac ester derivatives 1-gen-2007 Puglia, C.; Filosa, R.; Peduto, A.; De Caprariis, P.; Boatto, G.; Nieddu, M.; Santagati, N. A.; Bonina, F.
Molecular mechanism involved in the transport of a prodrug dopamine glycosyl conjugate 1-gen-2007 Dalpiaz, A.; Filosa, R.; de Caprariis, P.; Conte, G.; Bortolotti, F.; Biondi, C.; Scatturin, A.; Prasad, P. D.; Pavan, B.
Antioxidant activity of diphenylpropionamide derivatives: Synthesis, biological evaluation and computational analysis 1-gen-2008 Urbani, P.; Ramunno, A.; Filosa, R.; Pinto, A.; Popolo, A.; Bianchino, E.; Piotto, S.; Saturnino, C.; De Prisco, R.; Nicolaus, B.; Tommonaro, G.
Design, synthesis and biological evaluation of novel bicyclo[1.1.1]pentane-based ω-acidic amino acids as glutamate receptors ligands 1-gen-2009 Filosa, R.; Carmela Fulco, M.; Marinozzi, M.; Giacche, N.; Macchiarulo, A.; Peduto, A.; Massa, A.; de Caprariis, P.; Thomsen, C.; Christoffersen, C. T.; Pellicciari, R.
A new approach to di- And tetrasubstituted 2,3-dihydropyridin-4(1H)-ones through aza-diels-alder reaction promoted by silicon tetrachloride 1-gen-2009 Massa, A.; De Sio, V.; Villano, R.; Acocella, M. R.; Palombi, L.; Sellitto, G.; Peduto, A.; Filosa, R.; De Capraris, P.; Scettri, A.
Molecular modelling studies, synthesis and biological activity of a series of novel bisnaphthalimides and their development as new DNA topoisomerase II inhibitors 1-gen-2009 Filosa, R.; Peduto, A.; Di Micco, S.; Caprariis, P. d.; Festa, M.; Petrella, A.; Capranico, G.; Bifulco, G.
Synthesis of β-hydroxymalonates: the direct aldol addition of malonates to aldehydes in the presence of SiCl4 and i-Pr2EtN 1-gen-2009 Massa, A.; Scettri, A.; Filosa, R.; Capozzolo, L.
Trimethylchlorosilane and silicon tetrachloride in two novel methodologies for the efficient and mild aldol addition of β-keto esters and malonates to aldehydes 1-gen-2010 Massa, A.; Roscigno, A.; De Caprariis, P.; Filosa, R.; Di Mola, A.
Multi-component, regio-selective aldol addition of β-ketoesters to aldehydes: Scope and applications 1-gen-2011 More, V.; Di Mola, A.; Croce, G.; Tedesco, C.; Petronzi, C.; Peduto, A.; De Caprariis, P.; Filosa, R.; Massa, A.
Synthesis and cytotoxic activity of new β-carboline derivatives 1-gen-2011 Peduto, A.; More, V.; de Caprariis, P.; Festa, M.; Capasso, A.; Piacente, S.; de Martino, L.; de Feo, V.; Filosa, R.
The aldol addition of readily enolizable 1,3-dicarbonyl compounds to 2-cyanobenzaldehyde in the synthesis of novel 3-substituted isoindolinones 1-gen-2011 More, V.; Dimola, A.; Perillo, M.; Decaprariis, P.; Filosa, R.; Peduto, A.; Massa, A.
2,3-dihydro-1,2-diphenyl-substituted 4H-pyridinone derivatives as new anti flaviviridae inhibitors 1-gen-2011 Peduto, A.; Massa, A.; Di Mola, A.; de Caprariis, P.; La Colla, P.; Loddo, R.; Altamura, S.; Maga, G.; Filosa, R.
Structure-based design, synthesis and preliminary anti-inflammatory activity of bolinaquinone analogues 1-gen-2011 Petronzi, C.; Filosa, R.; Peduto, A.; Monti, M. C.; Margarucci, L.; Massa, A.; Ercolino, S. F.; Bizzarro, V.; Parente, L.; Riccio, R.; De Caprariis, P.
Design, synthesis, biophysical and biological studies of trisubstituted naphthalimides as G-quadruplex ligands 1-gen-2011 Peduto, A.; Pagano, B.; Petronzi, C.; Massa, A.; Esposito, V.; Virgilio, A.; Paduano, F.; Trapasso, F.; Fiorito, F.; Florio, S.; Giancola, C.; Galeone, A.; Filosa, R.
Mostrati risultati da 1 a 20 di 91
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